IPAM

Ipamorelin

A synthetic pentapeptide with the sequence Aib-His-D-2-Nal-D-Phe-Lys-NH2. It binds the growth hormone secretagogue receptor type 1a, the same receptor the endogenous peptide ghrelin acts on, and is described in the literature as selective for that receptor rather than acting across the wider set of pituitary secretagogue targets.

Ipamorelin has 2 registered human studies on ClinicalTrials.gov, reaching phase 2, covering 437 planned or enrolled participants across the 2 studies that published a figure. No FDA-approved product contains Ipamorelin. 18 papers naming it were published in the last ten years.

Collected 2026-08-02 from ClinicalTrials.gov and Drugs@FDA. Counts include only trials whose registered intervention names Ipamorelin; the registry search is fuzzy, so every match is re-checked. None of this says whether Ipamorelin works or is safe.

FDA status

Research only

Human studies

2

Furthest phase

Phase 2

Papers, 10 yr

18

Readership

6,559

monthly average, Feb–Jun 2026

Tracking since 2026-07-29 · About this data

What has actually been tested in humans

C

Phase 1 or 2 only

2

Registered human studies

Phase 2

Furthest phase reached

437

Planned or enrolled participants, across 2 studies that published a figure

None

No FDA-approved product contains it

3 loose registry matches were checked and 2 confirmed — 1 named something else and were discarded. We count a study only when Ipamorelin is named as an intervention in it.

Registered means registered — not that the study finished, and not that it found anything. The grade is mechanical: it is computed from the registry and the FDA record alone, and it grades how much is known, never whether a compound is good or safe. Collected 2026-08-02 from ClinicalTrials.gov and Drugs@FDA. Check the query.

What Ipamorelin is, and what it has been studied for

Ipamorelin is classified by ChEMBL as a protein, and appears in trial registrations under NNC 26-0161 and NNC-26-0161. Its FDA substance identifier is Y9M3S784Z6.

Across 2 registered trials, it has been studied in Ileus and Gastrointestinal Dysmotility. A condition here is what a sponsor registered the trial under — it records what was investigated, not what was shown.

The trials were run by Helsinn Therapeutics (U.S.), Inc. A named commercial sponsor means a compound is in formal development; its absence does not mean the opposite, only that no company has registered a trial under its own name.

How far it got

Ipamorelin reached Phase 2 across 2 registered trials.Phase 1First given to peoplePhase 2Looking for an effectPhase 3Tested at scalePhase 4Studied after approval

Ipamorelin reached Phase 2 across 2 registered trials.

No FDA-approved product contains Ipamorelin. A compound can stop at any rung for commercial reasons as easily as scientific ones, and the registry does not record which.

Is anyone studying Ipamorelin?

Papers published each year that name Ipamorelin in the title or abstract, with the clinical trials that started in the same year marked beneath. Ten calendar years.

03581017181920212223242526
Vertical axis: papers published that year. Bar for 2026 is hatched because that year is still running.
Publications and trials naming Ipamorelin, by year
YearPublicationsTrials startedComplete year
201720Yes
201840Yes
201910Yes
202020Yes
202100Yes
202200Yes
202300Yes
202420Yes
202500Yes
202680No

18 papers between 2017 and 2026. A paper counts when “Ipamorelin” appears in its title or abstract — phrase-matched, so a paper mentioning the words separately is not counted. The total is a single query over the whole window, which is why it does not equal the bars added together: PubMed files a paper under both its electronic and its print publication date, so one paper can appear in two years. Publication volume measures scientific attention, not whether a compound works: a well-studied compound can be well-studied and ineffective. Sources: PubMed and ClinicalTrials.gov · collected 2026-08-02.

Published research on Ipamorelin

18 indexed papers name Ipamorelin in their title or abstract. These are the 8 PubMed ranks most relevant. Listing a paper is not a judgement about it, and none of these is summarised here — follow the link and read what it says.

  1. Ipamorelin, the first selective growth hormone secretagogue

    Raun K, Hansen BS, Johansen NL, et al.European journal of endocrinology1998

    PMID 984982210.1530/eje.0.1390552

  2. Therapeutic Peptides in Orthopaedics: Applications, Challenges, and Future Directions

    Rahman OF, Lee SJ, Seeds WAJournal of the American Academy of Orthopaedic Surgeons. Global research & reviews2026

    PMID 4149020010.5435/JAAOSGlobal-D-25-00236

  3. Injectable Peptide Therapy: A Primer for Orthopaedic and Sports Medicine Physicians

    Mayfield CK, Bolia IK, Feingold CL, et al.The American journal of sports medicine2026

    PMID 4147642410.1177/03635465251357593

  4. Safety and Efficacy of Approved and Unapproved Peptide Therapies for Musculoskeletal Injuries and Athletic Performance

    Mendias CL, Awan TMSports medicine (Auckland, N.Z.)2026

    PMID 4196663910.1007/s40279-026-02437-0

  5. Beyond the androgen receptor: the role of growth hormone secretagogues in the modern management of body composition in hypogonadal males

    Sinha DK, Balasubramanian A, Tatem AJ, et al.Translational andrology and urology2020

    PMID 3225785510.21037/tau.2019.11.30

  6. Therapeutic Peptides in Aesthetic, Metabolic and Endocrine Conditions: Effects, Safety, Clinical Applications, and Future Perspectives

    Renke G, Chinellato LInternational journal of molecular sciences2026

    PMID 4212347110.3390/ijms27093890

  7. The growth hormone secretagogue receptor 1a agonists, anamorelin and ipamorelin, inhibit cisplatin-induced weight loss in ferrets: Anamorelin also exhibits anti-emetic effects via a central mechanism

    Lu Z, Ngan MP, Liu JYH, et al.Physiology & behavior2024

    PMID 3904335710.1016/j.physbeh.2024.114644

  8. Ipamorelin, a new growth-hormone-releasing peptide, induces longitudinal bone growth in rats

    Johansen PB, Nowak J, Skjaerbaek C, et al.Growth hormone & IGF research : official journal of the Growth Hormone Research Society and the International IGF Research Society1999

    PMID 1037334310.1054/ghir.1999.9998

Collected 2026-08-02from PubMed, phrase-matched on “Ipamorelin” in title and abstract. Run the same search.

About Ipamorelin

A synthetic pentapeptide with the sequence Aib-His-D-2-Nal-D-Phe-Lys-NH2. It binds the growth hormone secretagogue receptor type 1a, the same receptor the endogenous peptide ghrelin acts on, and is described in the literature as selective for that receptor rather than acting across the wider set of pituitary secretagogue targets.

Structure and mechanism only. Nothing above describes what this compound is for, and no dose appears anywhere on this page.

Reading on this compound

All articles

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